ALEXIS Biochemicals: Arachidonoyl cyclopropylamide

ALX-340-054

Revised 09-Jul-08

Arachidonoyl cyclopropylamide
SYNONYMS	ACPA N-Cyclopropyl-5Z,8Z,11Z,14Z-eicosatetraenamide
PRODUCT LINE	Neurobiology
PRODUCT CATEGORY	Anandamide & Anandamide Analogs

Ordering Information

Product Numbers:	Format:	Size:	Unit Price:	Quantity:	Add To Cart
ALX-340-054-M005		5 mg	46.00 USD

Product Specification

FORMULA:	C₂₃H₃₇NO
MW:	343.6
CAS NUMBER:	229021-64-1
PURITY:	≥98%
FORMULATION:	Liquid. Solution in ethanol.
SOLUBILITY:	10mg/ml soluble in 100% ethanol, DMSO or dimethyl formamide; 1mg/ml soluble in a 1:1 solution of in ethanol:PBS (pH 7.2) (dilute the ethanol solution with PBS).
SHIPPING:	SHIPPED ON BLUE ICE
LONG TERM STORAGE:	-20°C
USE/STABILITY:	Stable for at least 1 year after receipt when stored at -20°C. We do not recommend storing aqueous solutions for more than one day.

Product Description

Potent and selective CB₁ agonist (K_i=2.2nM). Displays 325-fold selectivity over CB₂ receptors (K_i=0.7µM). Active in vivo.

Product Specific Literature References

Synthesis and characterization of potent and selective agonists of the neuronal cannabinoid receptor (CB1): C.J. Hillard, et al.; J. Pharmacol. Exp. Ther. 289, 1427 (1999) Abstract
Arachidonylcyclopropylamide increases microglial cell migration through cannabinoid CB2 and abnormal-cannabidiol-sensitive receptors: A. Franklin, et al.; Eur. J. Pharmacol. 474, 195 (2003) Abstract
The interaction of cannabinoids and opioids on pentylenetetrazole-induced seizure threshold in mice: H. Shafaroodi, et al.; Neuropharmacology 47, 390 (2004) Abstract

General Information

BACKGROUND/TECHNICAL INFORMATION

To change the solvent, evaporate the ethanol under a gentle stream of nitrogen and immediately add the solvent of choice.

Further Categories Containing This Product:

Cannabinoid Receptor Agonists & Antagonists / Related Products

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