ALEXIS Biochemicals: ETB-Receptor Antagonist . sodium salt

ALX-155-020

Revised 17-Mar-08

ETB-Receptor Antagonist . sodium salt
SYNONYMS	BQ-788 . Na
PRODUCT LINE	Signal Transduction
PRODUCT CATEGORY	Endothelins [ETs] & Endothelin Receptors / Related Products

Ordering Information

Product Numbers:	Format:	Size:	Unit Price:	Quantity:	Add To Cart
ALX-155-020-MC05		0.5 mg	133.00 USD
ALX-155-020-M001		1 mg	185.00 USD

Product Specification

SEQUENCE:	N-cis-2,6-Dimethylpiperidinocarbonyl-L-γMeLeu-D-Trp(COOMe)-D-Nle-ONa
FORMULA:	C₃₄H₅₀N₅O₇Na
MW:	663.7
PEPTIDE CONTENT:	75-95%
PURITY:	≥95% (HPLC)
APPEARANCE:	White to off-white powder.
SOLUBILITY:	Soluble in methanol (0.5mg/ml), DMSO (4mg/ml), 0.1M sodium bicarbonate (3mg/ml) or 100% ethanol (4mg/ml); insoluble in water.
SHIPPING:	AMBIENT
LONG TERM STORAGE:	-20°C

Product Description

Highly potent and selective ET_B-receptor antagonist.

Product Specific Literature References

Clearance of circulating endothelin-1 by ETB receptors in rats: T. Fukuroda, et al.; BBRC 199, 1461 (1994) Abstract
Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788: K. Ishikawa, et al.; PNAS 91, 4892 (1994) Abstract

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