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Pyripyropenes, novel inhibitors of acyl-CoA:cholesterol acyltransferase produced by Aspergillus fumigatus. II. Structure elucidation of pyripyropenes A, B, C and D: Y.K. Kim, et al.; J. Antibiot. 47, 154 (1994) Abstract
Aflavinines and other antiinsectan metabolites from the ascostromata of Eupenicillium crustaceum and related species: H.J. Wang, et al.; Appl. Environ. Microbiol. 61, 4429 (1995) Abstract; Full Text
Total Synthesis of (+)-Pyripyropene A, a Potent, Orally Bioavailable Inhibitor of
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Biosynthesis of Pyripyropene A: H. Tomoda, et al.; J. Org. Chem. 61, 882 (1996)
Meroterpenoids with various biological activities produced by fungi: K. Shiomi, et al.; Pure Appl. Chem. 71, 1059 (1999) Full Text
A formal synthesis of (+)-pyripyropene A using a biomimetic epoxy-olefin cyclisation: effect of epoxy alcohol/ether on cyclisation efficiency: V.K. Aggarwal, et al.; J. Chem. Soc. 3315 (1999) Full Text
Mass-production of human ACAT-1 and ACAT-2 to screen isoform-specific inhibitor: a different substrate specificity and inhibitory regulation: K.H. Cho, et al.; BBRC 309, 864 (2003) Abstract
Identification of ACAT1- and ACAT2-specific inhibitors using a novel, cell-based fluorescence assay: individual ACAT uniqueness: A.T. Lada, et al.; J. Lipid Res. 45, 378 (2004) Abstract; Full Text
ACAT2 is localized to hepatocytes and is the major cholesterol-esterifying enzyme in human liver: P. Parini, et al.; Circulation 110, 2017 (2004) Abstract; Full Text
Exploiting PdII and TiIII chemistry to obtain gamma-dioxygenated terpenoids: synthesis of rostratone and novel approaches to aphidicolin and pyripyropene A: J. Justicia, et al.; J. Org. Chem. 70, 8265 (2005) Abstract
Total synthesis of alpha-pyrone meroterpenoids, novel bioactive microbial metabolites: T. Sunazuka and S. Omura; Chem. Rev. 105, 4559 (2005) Abstract
Potential therapeutics for obesity and atherosclerosis: inhibitors of neutral lipid metabolism from microorganisms: H. Tomoda & S. Omura; Pharmacol. Ther. 115, 375 (2007) Abstract
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