Synthesis and evaluation of phorboid 20-homovanillates: discovery of a class of ligands binding to the vanilloid (capsaicin) receptor with different degrees of cooperativity: G. Appendino, et al.; J. Med. Chem. 39, 3123 (1996) Abstract
A novel agonist, phorbol 12-phenylacetate 13-acetate 20-homovanillate, abolishes positive cooperativity of binding by the vanilloid receptor: A. Szallasi, et al.; Eur. J. Pharmacol. 299, 221 (1996) Abstract
A non-pungent resiniferatoxin analogue, phorbol 12-phenylacetate 13 acetate 20-homovanillate, reveals vanilloid receptor subtypes on rat trigeminal ganglion neurons: L. Liu, et al.; Neuroscience 84, 569 (1998) Abstract
Functional and desensitizing effects of the novel synthetic vanilloid- like agent 12-phenylacetate 13-acetate 20-homovanillate (PPAHV) in the perfused rat hindlimb: C.D. Griffiths, et al.; Br. J. Pharmacol. 131, 1408 (2000) Abstract
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology: J.C. Jerman, et al.; Br. J. Pharmacol. 130, 916 (2000) Abstract
Phorboid 20-homovanillates induce apoptosis through a VR1-independent mechanism: A. Macho, et al.; Chem. Biol. 7, 483 (2000) Abstract
Pharmacological differences between the human and rat vanilloid receptor 1 (VR1): P. McIntyre, et al.; Br. J. Pharmacol. 132, 1084 (2001) Abstract
Differences in sensitivity of vanilloid receptor 1 transfected to human embryonic kidney cells and capsaicin-activated channels in cultured rat dorsal root ganglion neurons to capsaicin receptor agonists: J.S. Shin, et al.; Neurosci. Lett. 299, 135 (2001) Abstract
Respiratory actions of vanilloid receptor agonists in the nucleus of the solitary tract: comparison of resiniferatoxin with non-pungent agents and anandamide: D.P. Geraghty, et al.; Br. J. Pharmacol. 137, 919 (2002) Abstract
Identification of species-specific determinants of the action of the antagonist capsazepine and the agonist PPAHV on TRPV1: E. Phillips, et al.; J. Biol. Chem. 279, 17165 (2004) Abstract
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