ALEXIS Biochemicals: nor-Binaltorphimine . dihydrochloride

ALX-550-111

Revised 12-May-03

nor-Binaltorphimine . dihydrochloride
SYNONYMS	nor-BNI . 2HCl
PRODUCT LINE	Neurobiology
PRODUCT CATEGORY	Opioid Receptors / Related Products

Ordering Information

Product Numbers:	Format:	Size:	Unit Price:	Quantity:	Add To Cart
ALX-550-111-M001		1 mg	25.00 USD

Product Specification

FORMULA:	C₄₀H₄₃N₃O₆ . 2HCl
MW:	661.8 . 73.0
CAS NUMBER:	105618-26-6
PURITY:	≥96%
APPEARANCE:	Tan solid.
SOLUBILITY:	Soluble in ethanol; sonification required.
SHIPPING:	AMBIENT
LONG TERM STORAGE:	-20°C
USE/STABILITY:	Aqueous solutions are highly unstable and should be freshly prepared.

Product Description

Highly selective κ-opioid receptor antagonist.

Product Specific Literature References

Binaltorphimine and nor-binaltorphimine, potent and selective kappa- opioid receptor antagonists: P.S. Portoghese, et al.; Life Sci. 40, 1287 (1987) Abstract
Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays: A.E. Takemori, et al.; J. Pharmacol. Exp. Ther. 246, 255 (1988) Abstract
Effects of the selective kappa opioid antagonist, nor-binaltorphimine, on electrically-elicited feeding in the rat: K.D. Carr, et al.; Life Sci. 45, 1787 (1989) Abstract
Structure-activity relationship of N17'-substituted norbinaltorphimine congeners. Role of the N17' basic group in the interaction with a putative address subsite on the kappa opioid receptor: P.S. Portoghese, et al.; J. Med. Chem. 37, 1495 (1994) Abstract
Differential agonist regulation of the human kappa-opioid receptor: A.D. Blake, et al.; J. Neurochem. 68, 1846 (1997) Abstract

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